Engineering and Improving Anti–CTLA-4 Checkpoint Inhibitors

Galvez-Cancino F., Parkes EE., Withers DR., Melero I.

Summary Next-generation anti–CTLA-4 antibodies have been designed and tested to improve the efficacy and therapeutic index by leveraging enhanced Fc-mediated effector function with conditional tumor-restricted activation. The goal is to achieve robust antitumor activity without inducing systemic immune-related toxicity. See related article by Jhatakia et al., p. 3289

DOI

10.1158/1078-0432.ccr-26-1059

Type

Journal article

Publisher

American Association for Cancer Research (AACR)

Publication Date

2026-08-03T00:00:00+00:00

Volume

32

Pages

3112 - 3114

Total pages

2

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