Synthesis and Biological Investigation of (+)-JD1, an Organometallic BET Bromodomain Inhibitor

Hassell-Hart S., Runcie A., Krojer T., Doyle J., Lineham E., Ocasio CA., Neto BAD., Fedorov O., Marsh G., Maple H., Felix R., Banks R., Ciulli A., Picaud S., Filippakopoulos P., von Delft F., Brennan PE., Stewart HJS., Chevassut TJ., Walker M., Austin C., Morley S., Spencer J.

DOI

10.1021/acs.organomet.9b00750

Type

Journal article

Journal

ORGANOMETALLICS

Publication Date

10/02/2020

Volume

39

Pages

408 - 416

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