Design, Synthesis and Characterization of Covalent KDM5 Inhibitors

Vazquez‐Rodriguez S., Wright M., Rogers CM., Cribbs AP., Velupillai S., Philpott M., Lee H., Dunford JE., Huber KVM., Robers MB., Vasta JD., Thezenas M., Bonham S., Kessler B., Bennett J., Fedorov O., Raynaud F., Donovan A., Blagg J., Bavetsias V., Oppermann U., Bountra C., Kawamura A., Brennan PE.

DOI

10.1002/anie.201810179

Type

Journal article

Journal

Angewandte Chemie International Edition

Publisher

Wiley

Publication Date

08/01/2019

Volume

58

Pages

515 - 519

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