Evaluation of linker length effects on a BET bromodomain probe
Traquete R., Henderson E., Picaud S., Cal PMSD., Sieglitz F., Rodrigues T., Oliveira R., Filippakopoulos P., Bernardes GJL.
A systematic study of the biological effects of introducing linkers of different chemical nature and length into BET bromodomain benzodiazepine ligands.