Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors
Lucas SCC., Atkinson SJ., Chung C-W., Davis R., Gordon L., Grandi P., Gray JJR., Grimes T., Phillipou A., Preston AG., Prinjha RK., Rioja I., Taylor S., Tomkinson NCO., Wall I., Watson RJ., Woolven J., Demont EH.