Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist

Balıkçı E., Marques A-SMC., Bauer LG., Seupel R., Bennett J., Raux B., Buchan K., Simelis K., Singh U., Rogers C., Ward J., Cheng C., Szommer T., Schützenhofer K., Elkins JM., Sloman DL., Ahel I., Fedorov O., Brennan PE., Huber KVM.

DOI

10.1021/acs.jmedchem.4c00072

Type

Journal article

Publisher

American Chemical Society (ACS)

Publication Date

2024-05-09T00:00:00+00:00

Volume

67

Pages

7245 - 7259

Total pages

14

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