Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors

Lucas SCC., Atkinson SJ., Chung C-W., Davis R., Gordon L., Grandi P., Gray JJR., Grimes T., Phillipou A., Preston AG., Prinjha RK., Rioja I., Taylor S., Tomkinson NCO., Wall I., Watson RJ., Woolven J., Demont EH.

DOI

10.1021/acs.jmedchem.1c00344

Type

Journal article

Journal

Journal of Medicinal Chemistry

Publisher

American Chemical Society (ACS)

Publication Date

12/08/2021

Volume

64

Pages

10711 - 10741

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