Design and synthesis of potent and selective inhibitors of BRD7 and BRD9 bromodomains
Hay DA., Rogers CM., Fedorov O., Tallant C., Martin S., Monteiro OP., Müller S., Knapp S., Schofield CJ., Brennan PE.
We describe potent and selective inhibitors of the BRD7 and BRD9 bromodomains intended for use as chemical probes to elucidate the biological roles of BRD7 and BRD9 in cells.