Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7

Gerken PA., Wolstenhulme JR., Tumber A., Hatch SB., Zhang Y., Müller S., Chandler SA., Mair B., Li F., Nijman SMB., Konietzny R., Szommer T., Yapp C., Fedorov O., Benesch JLP., Vedadi M., Kessler BM., Kawamura A., Brennan PE., Smith MD.

Original publication

DOI

10.1002/anie.201706788

Type

Journal article

Journal

Angewandte Chemie International Edition

Publisher

Wiley

Publication Date

04/12/2017

Volume

56

Pages

15555 - 15559