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Discovery of a Potent Dual SLK/STK10 Inhibitor Based on a Maleimide Scaffold.

Journal article

Serafim RAM. et al, (2021), Journal of medicinal chemistry

Structure-kinetic relationship reveals the mechanism of selectivity of FAK inhibitors over PYK2.

Journal article

Berger B-T. et al, (2021), Cell chemical biology

Aminothiazolones as potent, selective and cell active inhibitors of the PIM kinase family.

Journal article

Quevedo CE. et al, (2020), Bioorganic & medicinal chemistry, 28

Mining Public Domain Data to Develop Selective DYRK1A Inhibitors.

Journal article

Henderson SH. et al, (2020), ACS medicinal chemistry letters, 11, 1620 - 1626

Targeting the Water Network in Cyclin G-Associated Kinase (GAK) with 4-Anilino-quin(az)oline Inhibitors.

Journal article

Asquith CRM. et al, (2020), ChemMedChem, 15, 1200 - 1215

SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K.

Journal article

Wells C. et al, (2020), ACS medicinal chemistry letters, 11, 340 - 345

Development of 2-(4-pyridyl)-benzimidazoles as PKN2 chemical tools to probe cancer.

Journal article

Scott F. et al, (2020), Bioorganic & medicinal chemistry letters

Towards the Development of an In vivo Chemical Probe for Cyclin G Associated Kinase (GAK).

Journal article

Asquith CRM. et al, (2019), Molecules (Basel, Switzerland), 24

Development of Pyridine-based Inhibitors for the Human Vaccinia-related Kinases 1 and 2.

Journal article

Serafim RAM. et al, (2019), ACS Med Chem Lett, 10, 1266 - 1271

A Chemical Probe Targeting AAK1 and BMP2K

Journal article

Wells C. et al, (2019)

Structural mechanism of synergistic activation of Aurora kinase B/C by phosphorylated INCENP.

Journal article

Abdul Azeez KR. et al, (2019), Nature communications, 10

Crystal structure of human RIOK2 bound to a specific inhibitor.

Journal article

Wang J. et al, (2019), Open Biol, 9

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