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Frank N. et al, (2022), Nature, 611, 721 - 726
Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors
Journal article
Lucas SCC. et al, (2021), Journal of Medicinal Chemistry, 64, 10711 - 10741